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Novel Irreversible Inhibitors of Bruton's Tyrosine Kinase (BTK)
Invention Summary Bruton’s Tyrosine Kinase (BTK) is a nonreceptor cytoplasmic tyrosine kinase, predominantly expressed in hematopoietic cells. Targeted inhibition of BTK is a validated therapeutic strategy for diseases caused by abnormal activation of B-cells, including cancers, and autoimmune and inflammatory diseases. Drug discovery efforts...
Published: 7/16/2019   |   Inventor(s): David Bearss, Hariprasad Vankayalapati, Venkataswamy Sorna, Steven Warner, Sunil Sharma
Keywords(s):  
Category(s): Therapeutics, Small Molecule
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