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Novel Irreversible Inhibitors of Bruton's Tyrosine Kinase (BTK)
Invention Summary Bruton’s Tyrosine Kinase (BTK) is a nonreceptor cytoplasmic tyrosine kinase, predominantly expressed in hematopoietic cells. Targeted inhibition of BTK is a validated therapeutic strategy for diseases caused by abnormal activation of B-cells, including cancers, and autoimmune and inflammatory diseases. Drug discovery efforts...
Published: 7/16/2019
|
Inventor(s):
David Bearss
,
Hariprasad Vankayalapati
,
Venkataswamy Sorna
,
Steven Warner
,
Sunil Sharma
Keywords(s):
Category(s):
Therapeutics
,
Small Molecule
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